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Oncology & Targeted Therapies

Targeted oncology agents and precision therapeutics for clinical and translational research.

Erdafitinib

CAS 1346242-81-6

FGFR inhibitor

Pemigatinib

CAS 1503315-51-2

FGFR2 inhibitor

Futibatinib

CAS 1448428-04-3

FGFR inhibitor, irreversible

Infigratinib

CAS 872511-34-7

FGFR inhibitor

Rogaratinib

CAS 1443702-98-6

FGFR inhibitor

ASP5878

CAS 1453208-66-6

FGFR inhibitor

Dabogratinib (TYRA-300)

CAS 2800223-30-5

FGFR3 inhibitor

Vepugratinib (LOXO-435)

CAS 2833703-74-3

FGFR3 inhibitor

Lorlatinib

CAS 1454846-35-5

ALK inhibitor

Osimertinib

CAS 1421373-65-0

EGFR inhibitor

Gefitinib

CAS 184475-35-2

EGFR inhibitor

Erlotinib Hydrochloride

CAS 183319-69-9

EGFR inhibitor

Afatinib

CAS 850140-72-6

ErbB family inhibitor

Alectinib

CAS 1256580-46-7

ALK inhibitor

Crizotinib

CAS 877399-52-5

ALK/ROS1 inhibitor

Brigatinib

CAS 1197953-54-0

ALK inhibitor

Ibrutinib

CAS 936563-96-1

BTK inhibitor

Acalabrutinib

CAS 1420477-60-6

BTK inhibitor

Zanubrutinib

CAS 1691249-45-2

BTK inhibitor

Olaparib

CAS 763113-22-0

PARP inhibitor

Niraparib

CAS 1038915-60-4

PARP inhibitor

Rucaparib

CAS 283173-50-2

PARP inhibitor

Ribociclib

CAS 1211441-98-3

CDK4/6 inhibitor

Palbociclib

CAS 571190-30-2

CDK4/6 inhibitor

Abemaciclib

CAS 1231929-97-7

CDK4/6 inhibitor

Trametinib

CAS 871700-17-3

MEK inhibitor

Cobimetinib

CAS 934660-93-2

MEK inhibitor

Selumetinib

CAS 606143-89-9

MEK inhibitor

Alpelisib

CAS 1217486-61-7

PI3K inhibitor

Copanlisib

CAS 1032568-63-0

PI3K inhibitor

Idelalisib

CAS 870281-82-6

PI3K inhibitor

Ruxolitinib

CAS 941678-49-5

JAK1/2 inhibitor

Tofacitinib

CAS 477600-75-2

JAK inhibitor

Fedratinib

CAS 936091-14-4

JAK2 inhibitor

Sotorasib

CAS 2252403-56-6

KRAS G12C inhibitor

Adagrasib

CAS 2296729-00-3

KRAS G12C inhibitor

Venetoclax

CAS 1257044-40-8

BCL-2 inhibitor

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